Mentolad 50 mg/ml (Trestolone Acetate) 10ml vial
Active ingredient: trestolone acetate
Type: Anabolic steroid (19-nortestosterone derivative)
Form: Injection
Carrier oil: sesame oil
Description:
Trestolone (7alpha-methyl-19-nortestosterone, MENT), or trestolone, was one of several 19-nortestosterone derivatives considered as a possible male contraceptive therapy due to its unique chemical properties. Initially, pharmaceutical companies combined progesterone with testosterone to produce a viable male contraceptive option due to progesterone's ability to suppress spermatogenesis. Trestolone is unable to bind to 5alpha-reductase and therefore cannot be converted to DHT, making it a perfect candidate for a male androgen contraceptive.
Theoretically, trestolone has a ratio of 2300-650, meaning it is 23 times more anabolic than testosterone and 6.5 times more androgenic as well. But a 1992 study in rats found that the anabolic potency of this drug is 10 times greater than that of testosterone, while being 12 times more suppressive on the HPTA.
The reason for this lies in the unique alpha-methyl group on carbon 7 of the molecule. This methyl group stands out below the steroid ring structure and sterically inhibits conversion to DHT. However, Trestolone can still undergo aromatization and other androgen-dependent functions, causing it to effectively act like testosterone in the body, despite being a derivative of 19-nortestosterone.
Trestolone has also been shown to have minimal affinity for progesterone and mineralocorticoid receptors, despite being a nandrolone derivative. Testosterone is an anabolic steroid that initiates a fairly strong increase in muscle mass, which also significantly increases the dynamics of the protein synthesis process in the body. Minors should not use this drug because it can cause an unnatural and highly accelerated sexual maturation process. Trestolone was initially created primarily as an androgen substitute; this synthetic (or artificial) steroid, considered quite strong, was used.
The medical uses of trestolone include, among others: contraceptive treatment, rapid bone loss, benign prostatic hyperplasia, prostate cancer, primary hypogonadism, cachexia (a disease involving the so-called muscle wasting syndrome), sarcopenia, induced anabolism, and typically male pattern baldness.
Effects:
Extremely anabolic compound, 10x to 23x greater than testosterone.
It is extremely powerful in helping users burn fat and build muscle.
Increased strength and muscle mass.
Does not bind to SHBG.
Does not convert to DHT.
No significant increases in hematocrit or hemoglobin.
Rapid effect.
Increased appetite.
Side effects:
Significant increase in systolic blood pressure.
Rapid conversion to estrogen.
Dry throat.
Excessive sweating.
Upset stomach.
Diarrhea.
Heartburn.
Back acne.
Insomnia.
Night sweats
. Mood swings.
It is strongly recommended that an aromatase inhibitor such as Arimidex or letrozole be used when taking trestolone.
Your appetite should be extremely high and you will see a slight increase in gym strength. 1.25 mg of letrozole every other day to combat conversion to 7α-methylestradiol.
Dosage
: Beginner: 100 mg per week;
Intermediate: 200 mg per week;
Advanced: 300 mg per week.
It is advisable to start by taking 100 mg of trestolone acetate per week to see how your body responds. If your body responds well, you can consider increasing the dosage slowly, up to 300 mg per week.
Contraindications:
Pregnancy;
Known or suspected prostate or breast carcinoma;
Breastfeeding;
Hypersensitivity to the active substance or to any of the excipients;
High blood calcium levels.
Storage instructions:
Keep out of reach of children.
Store in a cool, dry place away from direct sunlight.
Store at room temperature.
Do not use after the expiration date.
Active ingredient: trestolone acetate
Type: Anabolic steroid (19-nortestosterone derivative)
Form: Injection
Carrier oil: sesame oil
Description:
Trestolone (7alpha-methyl-19-nortestosterone, MENT), or trestolone, was one of several 19-nortestosterone derivatives considered as a possible male contraceptive therapy due to its unique chemical properties. Initially, pharmaceutical companies combined progesterone with testosterone to produce a viable male contraceptive option due to progesterone's ability to suppress spermatogenesis. Trestolone is unable to bind to 5alpha-reductase and therefore cannot be converted to DHT, making it a perfect candidate for a male androgen contraceptive.
Theoretically, trestolone has a ratio of 2300-650, meaning it is 23 times more anabolic than testosterone and 6.5 times more androgenic as well. But a 1992 study in rats found that the anabolic potency of this drug is 10 times greater than that of testosterone, while being 12 times more suppressive on the HPTA.
The reason for this lies in the unique alpha-methyl group on carbon 7 of the molecule. This methyl group stands out below the steroid ring structure and sterically inhibits conversion to DHT. However, Trestolone can still undergo aromatization and other androgen-dependent functions, causing it to effectively act like testosterone in the body, despite being a derivative of 19-nortestosterone.
Trestolone has also been shown to have minimal affinity for progesterone and mineralocorticoid receptors, despite being a nandrolone derivative. Testosterone is an anabolic steroid that initiates a fairly strong increase in muscle mass, which also significantly increases the dynamics of the protein synthesis process in the body. Minors should not use this drug because it can cause an unnatural and highly accelerated sexual maturation process. Trestolone was initially created primarily as an androgen substitute; this synthetic (or artificial) steroid, considered quite strong, was used.
The medical uses of trestolone include, among others: contraceptive treatment, rapid bone loss, benign prostatic hyperplasia, prostate cancer, primary hypogonadism, cachexia (a disease involving the so-called muscle wasting syndrome), sarcopenia, induced anabolism, and typically male pattern baldness.
Effects:
Extremely anabolic compound, 10x to 23x greater than testosterone.
It is extremely powerful in helping users burn fat and build muscle.
Increased strength and muscle mass.
Does not bind to SHBG.
Does not convert to DHT.
No significant increases in hematocrit or hemoglobin.
Rapid effect.
Increased appetite.
Side effects:
Significant increase in systolic blood pressure.
Rapid conversion to estrogen.
Dry throat.
Excessive sweating.
Upset stomach.
Diarrhea.
Heartburn.
Back acne.
Insomnia.
Night sweats
. Mood swings.
It is strongly recommended that an aromatase inhibitor such as Arimidex or letrozole be used when taking trestolone.
Your appetite should be extremely high and you will see a slight increase in gym strength. 1.25 mg of letrozole every other day to combat conversion to 7α-methylestradiol.
Dosage
: Beginner: 100 mg per week;
Intermediate: 200 mg per week;
Advanced: 300 mg per week.
It is advisable to start by taking 100 mg of trestolone acetate per week to see how your body responds. If your body responds well, you can consider increasing the dosage slowly, up to 300 mg per week.
Contraindications:
Pregnancy;
Known or suspected prostate or breast carcinoma;
Breastfeeding;
Hypersensitivity to the active substance or to any of the excipients;
High blood calcium levels.
Storage instructions:
Keep out of reach of children.
Store in a cool, dry place away from direct sunlight.
Store at room temperature.
Do not use after the expiration date.